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OMDM-2
OMDM-2 是一种有效选择性的，代谢稳定的 anandamide 细胞摄取 (ACU) 抑制剂，Ki 值为 3.0 μM。
OMDM-2 Chemical Structure
CAS No. : 616884-63-0
| 规格 | 价格 | 是否有货 | |
|---|---|---|---|
| 1 mg | ￥387 | 询问价格 & 货期 | |
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| 生物活性 |
OMDM-2 is a potent, selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 3.0 μM[1]. |
IC50 & Target |
Ki: 3.0 μM (anandamide cellular uptake)[1] |
|---|---|
| 体外研究 (In Vitro) |
OMDM-2 shows poor affinity for either CB1 (Ki=5.1 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively; OMDM-2 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50=10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1]. Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only. |
| 分子量 |
431.65 |
| Formula |
C27H45NO3 |
| CAS 号 |
616884-63-0 |
| 结构分类 |
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| 初始来源 |
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
| 纯度 & 产品资料 |
Data Sheet (520 KB) 产品使用指南 (1538 KB)
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| 参考文献 |
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