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Swertiajaponin (Synonyms: 日当药黄素) 纯度: 99.84%
Swertiajaponin 是一种酪氨酸酶抑制剂，与酪氨酸酶结合囊形成多个氢键和疏水相互作用，IC50 值为 43.47 μM。Swertiajaponin 还能通过抑制氧化应激介导的 MAPK/MITF 信号导致酪氨酸酶蛋白水平下降。Swertiajaponin 能抑制黑色素积累，具有较强的抗氧化活性。
Swertiajaponin Chemical Structure
CAS No. : 6980-25-2
| 规格 | 价格 | 是否有货 | 数量 |
|---|---|---|---|
| 1 mg | ￥800 | In-stock | |
| 5 mg | ￥2100 | In-stock | |
| 10 mg | ￥3400 | In-stock | |
| 50 mg | 询价 | ||
| 100 mg | 询价 |
* Please select Quantity before adding items.
Swertiajaponin 相关产品
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| 生物活性 |
Swertiajaponin is a tyrosinase inhibitor, forms multiple hydrogen bonds and hydrophobic interactions with the binding pocket of tyrosinase, with an IC50 of 43.47 μM. Swertiajaponin also inhibits oxidative stress-mediated MAPK/MITF signaling, leading to decrease in tyrosinase protein level. Swertiajaponin suppresses melanin accumulation and exhibits strong anti-oxidative activity[1]. |
IC50 & Target |
IC50: 43.47 μM (tyrosinase)[1] |
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| 分子量 |
462.40 |
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| Formula |
C22H22O11 |
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| CAS 号 |
6980-25-2 |
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| 性状 |
固体 |
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| 颜色 |
Light yellow to yellow |
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| 中文名称 |
日当药黄素 |
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| 结构分类 |
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| 初始来源 |
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
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| 储存方式 |
4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
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| 溶解性数据 |
In Vitro:
DMSO 中的溶解度 : 250 mg/mL (540.66 mM; 超声助溶; 吸湿的 DMSO 对产品的溶解度有显著影响，请使用新开封的 DMSO) 配制储备液
查看完整储备液配制表
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)
Concentration (start) × Volume (start) = Concentration (final) × Volume (final) This equation is commonly abbreviated as: C1V1 = C2V2
动物溶解方案计算器
请输入动物实验的基本信息：
给药剂量 mg/kg 动物的平均体重 g 每只动物的给药体积 μL 动物数量 只 由于实验过程有损耗，建议您多配一只动物的量
计算结果
工作液所需浓度 : mg/mL
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| 纯度 & 产品资料 |
纯度: 99.84%
Data Sheet (604 KB) SDS (393 KB)
COA (172 KB) HNMR (316 KB) LCMS (93 KB) 产品使用指南 (1538 KB) |
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| 参考文献 |
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