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1-Caffeoylquinic acid 纯度: 99.06%
1-Caffeoylquinic acid 1-咖啡酰奎宁酸是一种有效的 NF-κB 抑制剂,对 p105 的 RH 结构域显示高结合亲和力,Ki 值为 0.002 μM,结合能为 1.50 Kcal/mol。1-Caffeoylquinic acid 具有抗氧化应激能力。 1-Caffeoylquinic acid 抑制 PD-1/PD-L1 相互作用。
1-Caffeoylquinic acid Chemical Structure
CAS No. : 1241-87-8
规格 | 价格 | 是否有货 | 数量 |
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1 mg | ¥850 | In-stock | |
5 mg | ¥2100 | In-stock | |
10 mg | ¥3400 | In-stock | |
50 mg | 询价 | ||
100 mg | 询价 |
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1-Caffeoylquinic acid 相关产品
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生物活性 |
1-Caffeoylquinic acid is an effective NF-κB inhibitor, shows significant binding affinity to the RH domain of p105 with Ki of 0.002 μM and binding energy of 1.50 Kcal/mol[1]. 1-Caffeoylquinic acid has anti-oxidative stress ability[2]. 1-Caffeoylquinic acid inhibits PD-1/PD-L1 interact[3]. |
IC50 & Target |
Ki: 0.002 μM (1-Caffeoylquinic acid)[1] |
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分子量 |
354.31 |
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Formula |
C16H18O9 |
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CAS 号 |
1241-87-8 |
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性状 |
固体 |
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颜色 |
White to off-white |
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结构分类 |
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初始来源 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
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溶解性数据 |
In Vitro:
DMSO 中的溶解度 : 250 mg/mL (705.60 mM; 超声助溶; 吸湿的 DMSO 对产品的溶解度有显著影响,请使用新开封的 DMSO) 配制储备液
查看完整储备液配制表
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)
Concentration (start) × Volume (start) = Concentration (final) × Volume (final) This equation is commonly abbreviated as: C1V1 = C2V2
动物溶解方案计算器
请输入动物实验的基本信息:
给药剂量 mg/kg 动物的平均体重 g 每只动物的给药体积 μL 动物数量 只 由于实验过程有损耗,建议您多配一只动物的量
计算结果
工作液所需浓度 : mg/mL
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纯度 & 产品资料 |
纯度: 99.06%
Data Sheet (600 KB) SDS (251 KB)
COA (194 KB) HNMR (159 KB) RP-HPLC (326 KB) 产品使用指南 (1538 KB) |
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参考文献 |
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