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Myosmine (Synonyms: 麦斯明) 纯度: 99.95%
Myosmine 是存在于坚果和坚果制品中的特定烟草生物碱，对 a4b2 烟碱乙酰胆碱受体 ( nAChR) 具有低亲和力，Ki 值为 3300 nM。
Myosmine Chemical Structure
CAS No. : 532-12-7
| 规格 | 价格 | 是否有货 | 数量 |
|---|---|---|---|
| Free Sample (0.1 – 0.2 mg) | Apply now | ||
| 10 mM * 1 mL in DMSO | ￥550 | In-stock | |
| 100 mg | ￥500 | In-stock | |
| 250 mg | ￥1000 | In-stock | |
| 500 mg | 询价 | ||
| 1 g | 询价 |
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Myosmine 相关产品
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| 生物活性 |
Myosmine, a specific tobacco alkaloid in nuts and nut products, has low affinity for a4b2 nicotinic acetylcholinergic receptors (nAChR) with a Ki of 3300 nM[1][2]. |
IC50 & Target |
Ki: 3300 nM (a4b2 nAChR) and >10 µM (AT1)[1] |
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| 体外研究 (In Vitro) |
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| 体内研究 (In Vivo) |
Myosmine (0.001, 0.005, 0.5, and 50 micromol/kg; oral; in Wistar rats) causes a higher percentage of the radioactivity excreted in urine (86.2% and 88.9%) at the two lower doses (0.001 and 0.005 micromol/kg),as compared with the higher doses (0.5 and 50 micromol/kg), where only 77.8% and 75.4% of the dose is found in urine[2]. Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only. |
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| 分子量 |
146.19 |
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| Formula |
C9H10N2 |
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| CAS 号 |
532-12-7 |
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| 性状 |
<42°C 固体,>44°C 液体 |
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| 颜色 |
Off-white to yellow |
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| 中文名称 |
麦斯明 |
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| 结构分类 |
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| 初始来源 |
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
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| 储存方式 |
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| 溶解性数据 |
In Vitro:
H2O 中的溶解度 : ≥ 100 mg/mL (684.04 mM) DMSO 中的溶解度 : 100 mg/mL (684.04 mM; 超声助溶; 吸湿的 DMSO 对产品的溶解度有显著影响，请使用新开封的 DMSO) * “≥” means soluble, but saturation unknown. 配制储备液
查看完整储备液配制表
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。 * 备注：如您选择水作为储备液，请稀释至工作液后，再用 0.22 μm 的滤膜过滤除菌后使用。
Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)
Concentration (start) × Volume (start) = Concentration (final) × Volume (final) This equation is commonly abbreviated as: C1V1 = C2V2
动物溶解方案计算器
请输入动物实验的基本信息：
给药剂量 mg/kg 动物的平均体重 g 每只动物的给药体积 μL 动物数量 只 由于实验过程有损耗，建议您多配一只动物的量
计算结果
工作液所需浓度 : mg/mL
该产品水溶性佳，请具体参考实测 水 / PBS / Saline 中的溶解度数据。
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| 纯度 & 产品资料 |
纯度: 99.95%
Data Sheet (601 KB) SDS (0 KB)
COA (195 KB) HNMR (119 KB) GC (191 KB) 产品使用指南 (1538 KB) |
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| 参考文献 |
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