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(R)-Mirtazapine D3(Synonyms: (R)-Org3770 D3; (R)-6-Azamianserin D3)

发表于由

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(R)-Mirtazapine D3 (Synonyms: (R)-Org3770 D3; (R)-6-Azamianserin D3)

(R)-Mirtazapine D3 ((R)-Org3770 D3) 是 (R)-Mirtazapine 氘代物。(R)-Mirtazapine 是 Mirtazapine 的 R(−)-对映异构体，在急性热伤害感受动物模型中具有抗伤害感受的作用。(R)-Mirtazapine 是 5-HT3 受体拮抗剂，在体内主要经 CYP3A4 代谢。

(R)-Mirtazapine D3(Synonyms: (R)-Org3770 D3; (R)-6-Azamianserin D3)

(R)-Mirtazapine D3 Chemical Structure

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生物活性

(R)-Mirtazapine D3 ((R)-Org3770 D3) is a deuterium labeled (R)-Mirtazapine. (R)-Mirtazapine is a R(−)-enantiomer of Mirtazapine with antinociceptive properties in an animal model of acute thermal nociception. (R)-Mirtazapine is a 5-HT3 receptor antagonist. (R)-Mirtazapine is mainly metabolized by CYP3A4[1].

IC50 & Target

5-HT3 Receptor

 

分子量

268.37

Formula

C17H16D3N3
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Muth-Selbach U, et al. Racemic intrathecal mirtazapine but not its enantiomers acts anti-neuropathic after chronic constriction injury in rats. Brain Res Bull. 2009 Apr 6;79(1):63-8.

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