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(S)-Mirtazapine D3(Synonyms: (S)-Org3770 D3; (S)-6-Azamianserin D3)

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(S)-Mirtazapine D3 (Synonyms: (S)-Org3770 D3; (S)-6-Azamianserin D3)

(S)-Mirtazapine D3 ((S)-Org3770 D3) 是 (S)-Mirtazapine 氘代物。(S)-Mirtazapine 是 Mirtazapine 的 S(+)-对映异构体，在急性热伤害感受动物模型中具有促伤害感受的特性。(S)-Mirtazapine 是一种立体选择性 5-HT2 受体拮抗剂，在体内被 CYP2D6 和 CYP1A2 代谢。

(S)-Mirtazapine D3(Synonyms: (S)-Org3770 D3; (S)-6-Azamianserin D3)

(S)-Mirtazapine D3 Chemical Structure

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生物活性

(S)-Mirtazapine D3 ((S)-Org3770 D3) is a deuterium labeled (S)-Mirtazapine. (S)-Mirtazapine is a S(+)-enantiomer of Mirtazapine with pronociceptive properties in an animal model of acute thermal nociception.(S)-Mirtazapine is a stereoselective 5-HT2 receptor antagonist. (S)-Mirtazapine is metabolized by CYP2D6 and CYP1A2[1].

IC50 & Target

5-HT2 receptor[1]
分子量

268.37

Formula

C17H16D3N3
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Muth-Selbach U, et al. Racemic intrathecal mirtazapine but not its enantiomers acts anti-neuropathic after chronic constriction injury in rats. Brain Res Bull. 2009 Apr 6;79(1):63-8.

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